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ici182780
释义
ici182780
雌激素拮抗剂,对雌激素依赖的乳腺癌细胞MCF-7荷瘤裸鼠的抑瘤率>80%,而在相同条件下,三苯氧胺的抑瘤率仅为40%。可阻止雌激素受体进入细胞核并可使该受体的总水平下降,使雌激素受体通路完全切断,三苯氧胺则不能完全阻断该受体通路,而只有部分拮抗作用。
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更新时间:2026/6/28 22:10:01